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NEUROSERVICE offers standardized tests revealing precise biological mechanisms, validating a target, allowing bench-mark with reference pharmacological tools or approved drugs.

Catalog of Pharmacological Tests:

CodeNameTargetPharm. Ref.BiologyDownload
P-001Fast sodium channel inhibitionSodium channelsTetrodotoxinAction Potential genesis and propagation
P-002AMPA-mediated synaptic transmissionAMPA/Kainate receptorsNBQXGlutamatergic synaptic transmission
P-003NMDA receptors competitive antagonistNMDA receptorsD-AP5Long-Term Potentiation
P-004GABA-A receptors - Network ExcitabilityGABA-A receptorsBicucullineEpileptiform activity
P-005Neurosteroids / GABA-A receptorsGABA-A receptorsGanaxoloneAllosteric modulation of GABA-A
P-006Inhibition of phasic GABA-A receptorsPhasic GABA-A receptorsGabazin (SR-95531)GABA-A receptor-mediated fast synaptic transmission
P-007DHPG - induced LTDmGluR1 & mGluR5 receptorsDHPGLTD induced by mGluR1/mGluR5 activation
P-008AMPA/kainate receptors-mediated excitotoxicityAMPA/kainate receptorskainateExcitotoxicity
P-009L-type calcium channels / Synaptic TransmissionL-type VDCCNifedipineModulation of synaptic transmission by VDCC
P-010Cholinergic transmission - Alzheimer's diseaseAcetylcholinesterasePhysostigmine (Eserine)cholinergic modulation of glutamate neurotransmission
P-011NMDA & nicotinic receptors / Alzheimer's & Parkinson's diseasesNMDA & nicotinic receptorsMemantineLong-Term Potentiation / Memory
P-012H3 histamine receptor-dependent depression in Dentate GyrusH3 histamine receptorR-alpha-methylhistaminePre-synaptic H3 receptor
P-013Histamine receptors mediated increase of CA1 pyramidal neurons firingH1 and H2 histamine receptorsHistamineCA1 pyramidal neurons spontaneous activity
P-014mGluR2-mediated depression of synaptic transmission at MPP synapsesmGluR2 receptorsDCG-IVpre-synaptic mGluR2 receptors
P-015dopamine-induced increase of synaptic transmission and plasticityD1/D5 dopamine receptorsSCH23390dopaminergic modulation of synaptic transmission
P-016Model of 4-AP-induced epilepsyK+ channelPhenytoin / CarbamazepineIn vitro epilepsy model
P-017Model of low-magnesium-induced epilepsyNMDA receptorPhenytoin / CarbamazepineIn vitro epilepsy model
P-018Model of bicuculline-induced epilepsyGABA-A receptorSomatostatinIn vitro model of epilepsy
P-019Model of cholinergic-induced epilepsyGABA-A / M1muscarinic receptorsdiazepamIn vitro epilepsy model

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